Collect. Czech. Chem. Commun. 1998, 63, 698-712
https://doi.org/10.1135/cccc19980698

Azachalcone Derivatives and Their Bis Substituted Analogs as Novel Antimycobacterial Agents

Václav Kozmíka, Pavel Lhotáka, Želmíra Odlerováb and Jaroslav Palečeka

a Department of Organic Chemistry, Prague Institute of Chemical Technology, 166 28 Prague 6, Czech Republic
b Institute of Preventive and Clinical Medicine, 833 01 Bratislava, Slovak Republic

Individual author index pages


Other CCCC articles of these authors

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    2004, Vol. 69, Issue 2, pp. 365–383 [Abstract]
  • Marie Mézlová, Hana Petříčková, Petr Maloň, Václav Kozmík and Jiří Svoboda*
    Axially Chiral 3,3'-Bi(1-benzothiophene)-2,2'-dicarboxylic Acid and Its Derivatives
    2003, Vol. 68, Issue 5, pp. 1020–1038 [Abstract]
  • Simon Cihelník, Ivan Stibor* and Pavel Lhoták
    Solvent-Free Synthesis of Sulfonephthaleins, Sulfonefluoresceins and Fluoresceins Under Microwave Irradiation
    2002, Vol. 67, Issue 12, pp. 1779–1789 [Abstract]
  • Bedřich Košata, Václav Kozmík and Jiří Svoboda*
    Reactivity of [1]Benzothieno[3,2-b][1]benzothiophene - Electrophilic and Metallation Reactions
    2002, Vol. 67, Issue 5, pp. 645–664 [Abstract]
  • Ivan Stibor*, Martina Růžičková, Rostislav Krátký, Michal Vindyš, Jaroslav Havlíček, Evguenni Pinkhassik, Pavel Lhoták, Asiya R. Mustafina, Yuliya E. Morozova, Ella Kh. Kazakova and Valentina P. Gubskaya
    New Calix[4]arene-Based Amides - Their Synthesis, Conformation, Complexation
    2001, Vol. 66, Issue 4, pp. 641–662 [Abstract]
  • Pavel Lhoták*, Václav Šťastný, Petra Zlatušková, Ivan Stibor, Veronika Michlová, Marcela Tkadlecová, Jaroslav Havlíček and Jan Sýkora
    Synthesis and 1H NMR Complexation Study of Thiacalix[4]arene Tetraacetates
    2000, Vol. 65, Issue 5, pp. 757–771 [Abstract]
  • Pavel Pihera, Jaroslav Paleček and Jiří Svoboda
    Diels-Alder Reactions of [1]Benzothieno[3,2-b]furan
    1998, Vol. 63, Issue 5, pp. 681–697 [Abstract]
  • Jiří Kuneš, Jiří Jáchym, Petr Jirásko, Želmíra Odlerová and Karel Waisser
    Combination of the Topliss Approach with the Free-Wilson Analysis in the Study of Antimycobacterial Activityof 4-Alkylthiobenzanilides
    1997, Vol. 62, Issue 9, pp. 1503–1510 [Abstract]
  • Miroslav Terinek, Václav Kozmík and Jaroslav Paleček
    Prostanoids: Synthesis of Enantiomers of 15-Deoxy-16-hydroxy-16-methylprostaglandin E1
    1997, Vol. 62, Issue 8, pp. 1325–1341 [Abstract]
  • Hans-Dietrich Stachel, Želmíra Odlerová and Karel Waisser
    A New Pharmacophore of Potential Antimycobacterial Activity: The Disulfide Group in the Ring of Alicyclic Compounds
    1997, Vol. 62, Issue 3, pp. 510–515 [Abstract]
  • Jiří Svoboda, Václav Kozmík, Ivan Veselý and Jaroslav Paleček
    New Synthesis of Important Prostanoid Intermediate
    1996, Vol. 61, Issue 10, pp. 1509–1519 [Abstract]
  • Jiří Hartl, Martin Doležal, Jana Krinková, Antonín Lyčka and Želmíra Odlerová
    Synthesis and Antituberculotic Activity of 5-Alkyl-6-chloro-2-pyrazinecarboxamides and Corresponding Thioamides
    1996, Vol. 61, Issue 7, pp. 1109–1114 [Abstract]
  • Martin Doležal, Jiří Hartl, Antonín Lyčka, Vladimír Buchta and Želmíra Odlerová
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    1996, Vol. 61, Issue 7, pp. 1102–1108 [Abstract]
  • Jiří Svoboda, Pavel Pihera, Petr Sedmera and Jaroslav Paleček
    Electrophilic Substitution Reactions of [1]Benzothieno[3,2-b]furan
    1996, Vol. 61, Issue 6, pp. 888–900 [Abstract]
  • Karel Waisser, Jiří Kuneš, Alexandr Hrabálek, Miloš Macháček and Želmíra Odlerová
    New Groups of Potential Antituberculotics: 5-Alkylthio-1-aryltetrazoles
    1996, Vol. 61, Issue 5, pp. 791–798 [Abstract]
  • Jiří Svoboda and Jaroslav Paleček
    New Method for Preparation of 1-Azabicyclo[2.2.2]octane-4-carbonitrile and 1-Azabicyclo[3.2.2]nonane-5-carbonitrile
    1995, Vol. 60, Issue 9, pp. 1536–1540 [Abstract]
  • Jaroslav Paleček and Ivan Veselý
    Synthesis of Monomeric 2-[(2-Methyl-2-propenoyl)oxy]ethyl Esters of Prostaglandins
    1995, Vol. 60, Issue 7, pp. 1242–1246 [Abstract]
  • Martin Doležal, Jiří Hartl, Antonín Lyčka, Vladimír Buchta and Želmíra Odlerová
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    1995, Vol. 60, Issue 7, pp. 1236–1241 [Abstract]
  • Václav Kozmík and Jaroslav Paleček
    Synthetic Analogues of 15,15-Acetals of Prostaglandin F2α and E2
    1994, Vol. 59, Issue 11, pp. 2533–2544 [Abstract]
  • Karel Waisser, Jiří Kuneš, Alexandr Hrabálek and Želmíra Odlerová
    New Groups of Potential Antituberculotics: Bis(1-aryltetrazol-5-yl) Disulfides. Structure Activity Relationship
    1994, Vol. 59, Issue 1, pp. 234–238 [Abstract]
  • Václav Kozmík and Jaroslav Paleček
    Synthetic Analogues of Prostaglandins F2α and E2
    1994, Vol. 59, Issue 1, pp. 138–148 [Abstract]
  • Jiří Svoboda, Miloslav Nič and Jaroslav Paleček
    Synthesis of [1]Benzothieno[3,2-b]furan - A New Fused Benzoheterocyclic System
    1993, Vol. 58, Issue 12, pp. 2983–2986 [Abstract]
  • Karel Waisser, Lenka Kubicová, Věra Klimešová and Želmíra Odlerová
    New Groups of Potential Antituberculotics: 3-Aryl-2H,4H-benz[e][1,3]oxazine-2,4-diones. Comparison of the Topliss Approach with Regression Analysis
    1993, Vol. 58, Issue 12, pp. 2977–2982 [Abstract]
  • Pavel Lhoták and Antonín Kurfürst
    Synthesis of Luminophoric Derivatives of PBD Based on 2,5-Diaryl Substituted Thiazoles and Oxazoles
    1993, Vol. 58, Issue 11, pp. 2720–2728 [Abstract]
  • Pavel Lhoták and Antonín Kurfürst
    Synthesis of Luminophores Based on Thiazole Derivatives of PBD
    1993, Vol. 58, Issue 8, pp. 1898–1904 [Abstract]
  • Jiří Svoboda, Miloslav Nič and Jaroslav Paleček
    Application of Magnesium Alkoxides to Syntheses of Benzoheterocyclic Compounds
    1993, Vol. 58, Issue 3, pp. 592–599 [Abstract]
  • Karel Waisser, Lenka Kubicová and Želmíra Odlerová
    Antituberculotic 4'-Cyclohexylthiobenzanilides: Combination of Free-Wilson Method in QSAR with Topliss Approach
    1993, Vol. 58, Issue 1, pp. 205–212 [Abstract]
  • Karel Waisser, Miloš Macháček, Želmíra Odlerová, Wilfried Thiel and Roland Mayer
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    1993, Vol. 58, Issue 1, pp. 197–204 [Abstract]
  • Karel Waisser, Jiří Kuneš, Jiří Klimeš, Miroslav Polášek and Želmíra Odlerová
    Relations between Structure and Antituberculotic Activity of 4-Alkoxybenzoic Acids
    1993, Vol. 58, Issue 1, pp. 191–196 [Abstract]
  • Pavel Lhoták and Antonín Kurfürst
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    1992, Vol. 57, Issue 9, pp. 1937–1946 [Abstract]
  • Václav Kozmík and Jaroslav Paleček
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    1992, Vol. 57, Issue 7, pp. 1483–1486 [Abstract]
  • Pavel Lhoták, Antonín Kurfürst and Petr Nádeník
    The Synthetic Use of 2-(4'-Acetylbiphenyl-4-yl)-5-phenyl-1,3,4-oxadiazole for Preparation of New Heterocyclic Luminophores
    1992, Vol. 57, Issue 2, pp. 385–392 [Abstract]
  • Richard Hrabal, Pavel Lhoták and Antonín Kurfürst
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    1992, Vol. 57, Issue 2, pp. 375–384 [Abstract]
  • Ivan Veselý, Jaroslav Paleček and Ivan Stibor
    Resolution of a Racemic Corey Lactone via Enantioselective Esterification
    1992, Vol. 57, Issue 2, pp. 357–361 [Abstract]
  • Jiří Svoboda, Miloslav Nič and Jaroslav Paleček
    An Anomalous Course of the Darzens Reaction Catalyzed with Magnesium Methoxide
    1992, Vol. 57, Issue 1, pp. 119–122 [Abstract]
  • Karel Waisser, Jiří Kuneš and Želmíra Odlerová
    Correlation of structural parameters with antituberculotic activity in a group of 2-benzamidobenzothiazoles
    1991, Vol. 56, Issue 12, pp. 2978–2985 [Abstract]
  • Bohumil Žák, Ivan Veselý, Karel Neumitka and Jaroslav Paleček
    Preparation of optically pure enatiomers of Corey lactone by resolution of the racemate
    1991, Vol. 56, Issue 8, pp. 1690–1700 [Abstract]
  • Antonín Kurfürst, Pavel Lhoták, Petr Nádeník, Františka Raclová-Pavlíková and Josef Kuthan
    2-(Biphenyl-4-yl)-5-phenyl-1,3,4-oxadiazole (PBD): Electrophilic 4’-substitution and following transformations
    1991, Vol. 56, Issue 7, pp. 1495–1504 [Abstract]
  • Jiří Svoboda and Jaroslav Paleček
    Synthesis of N-[(3-substituted phenoxy)alkyl]acetohydroxamic acids, potential inhibitors of the enzyme 5-lipoxygenase
    1991, Vol. 56, Issue 6, pp. 1317–1332 [Abstract]
  • Antonín Kurfürst, Josef Kuthan, Pavel Lhoták, Petr Nádeník, Werner Schroth and Roland Spitzner
    4-(5-Phenyl-1,3,4-oxadiazol-2-yl)biphenyl-4'-carboxylic acid: Its functional derivatives and their heterocyclization into 1,3-thiazine-6-thiones
    1990, Vol. 55, Issue 11, pp. 2722–2730 [Abstract]
  • Karel Dlabal, Karel Palát, Antonín Lyčka and Želmíra Odlerová
    Synthesis and 1H and 13C NMR spectra of sulfur derivatives of pyrazine derived from amidation product of 2-chloropyrazine and 6-chloro-2-pyrazinecarbonitrile. Tuberculostatic activity
    1990, Vol. 55, Issue 10, pp. 2493–2501 [Abstract]
  • Karel Waisser, Nestor Houngbedji, Miloš Macháček, Miroslav Sekera, Josef Urban and Želmíra Odlerová
    Antimycobacterial thiobenzanilides
    1990, Vol. 55, Issue 1, pp. 307–316 [Abstract]
  • Ivan Veselý, Václav Kozmík, Václav Dědek, Jaroslav Paleček, Jiří Mostecký and Ivan Stibor
    Large-scale synthesis of racemic “Corey lactone”
    1989, Vol. 54, Issue 6, pp. 1683–1686 [Abstract]
  • Antonín Kurfürst, Pavel Lhoták, Miroslav Petrů and Josef Kuthan
    Oligophenylene 2,4,6-triarylpyridines and analogous diaza-p-terphenyls, diaza-p-quaterphenyls and diaza-p-quinquephenyls with luminiscent activity
    1989, Vol. 54, Issue 2, pp. 462–472 [Abstract]
  • Jiří Svoboda, Zuzana Kocfeldová and Jaroslav Paleček
    Reaction of 4-substituted benzaldehydes and acetophenones with chloroacetonitrile
    1988, Vol. 53, Issue 4, pp. 822–832 [Abstract]
  • Jiří Svoboda, Karel Čapek and Jaroslav Paleček
    Esters of arylpropionic acids with 1,2:5,6-di-O-isopropylidene- and 1,2-O-isopropylidene-α-D-glucofuranose
    1987, Vol. 52, Issue 3, pp. 766–774 [Abstract]
  • Jiří Svoboda, Jaroslav Paleček and Václav Dědek
    Phase transfer catalysed N-substitution of 2H-1,2-benzisothiazolin-3-one 1,1-dioxide
    1986, Vol. 51, Issue 6, pp. 1304–1310 [Abstract]
  • Jiří Svoboda, Jaroslav Paleček and Václav Dědek
    The synthesis of substituted 2H-1,2-benzothiazines 1,1-dioxides
    1986, Vol. 51, Issue 5, pp. 1133–1139 [Abstract]
  • Jiří Svoboda, Jaroslav Paleček, Václav Dědek and Jiří Mostecký
    One-step synthesis of substituted 2-aryl-2-bromoalkyl-1,3-dioxolanes
    1984, Vol. 49, Issue 6, pp. 1515–1520 [Abstract]
  • Jaroslav Paleček, Manfred Pavlík and Josef Kuthan
    Chemical transformations of ethyl 3,5-dicyano-2,4,4,6-tetramethyl-1,4-dihydro-1-pyridyl acetate, sythesis of a new N-vinyl monomer
    1983, Vol. 48, Issue 2, pp. 617–622 [Abstract]
  • Jaroslav Paleček, Manfred Pavlík and Josef Kuthan
    N-alkylation of Hantzsch 1,4-dihydropyridines with esters of halogenocarboxylic acids
    1983, Vol. 48, Issue 2, pp. 608–616 [Abstract]
  • Josef Kuthan, Jaroslav Paleček and Jiří Valihrach
    Stable 2H-pyran derivatives accessible by cyclocondensation of p-substituted benzoylacetonitriles
    1981, Vol. 46, Issue 3, pp. 748–758 [Abstract]
  • Jaroslav Paleček, Jaroslav Kopecký and Josef Kuthan
    N-alkylation of 3,5-dicyano-2,4,4,6-tetramethyl-1,4-dihydropyridine with some α,ω-dihalogeno-N-alkenes
    1980, Vol. 45, Issue 12, pp. 3370–3377 [Abstract]
  • Josef Kuthan, Antonín Kurfürst, Zdeněk Prošek and Jaroslav Paleček
    Substituent effect in 1H-NMR spectra of the Hantzsch 1,4-dihydropyridines. meta and para Substituted 4-phenyl derivatives
    1978, Vol. 43, Issue 4, pp. 1068–1079 [Abstract]
  • Lubomír Musil, Jaroslav Paleček and Josef Kuthan
    Substituent effect in electronic and 1H-NMR spectra of 1- and 4-alkylated 3,5-dicyano-2,6-dimethyl-1,4-dihydropyridines
    1978, Vol. 43, Issue 4, pp. 946–959 [Abstract]
  • Vratislav Skála, Stanislav Böhm, Jaroslav Paleček and Josef Kuthan
    Electronic and mass spectra of 2,6-disubstituted phenyl and 2-styryl derivatives of 3,5-dicyanopyridines and their 1,4-dihydroanalogues
    1978, Vol. 43, Issue 2, pp. 434–446 [Abstract]