Collect. Czech. Chem. Commun. 1994, 59, 421-428
https://doi.org/10.1135/cccc19940421

The Deamino-Carba Analogs of Vasotocin. Synthesis and Some Biological Properties

Zdenko Procházkaa, Jiřina Slaninováa, Per Melinb, Carl-Johan Aurellb and Michal Lebla

a Institute of Organic Chemistry and Biochemistry, Academy of Sciences of the Czech Republic, 166 10 Prague 6, Czech Republic
b Ferring AB, Malmö, Sweden

Individual author index pages


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    Synthesis and properties of oxytocin analogues with high and selective natriuretic activity
    1982, Vol. 47, Issue 9, pp. 2540–2560 [Abstract]
  • Zdenko Procházka, Miloš Buděšínský, Jorga Smolíková, Petr Trška and Karel Jošt
    1-Aminocyclopropanecarboxylic acid and its derivatives
    1982, Vol. 47, Issue 8, pp. 2291–2305 [Abstract]
  • Jiřina Slaninová, Iain C. A. F. Robinson, Pavel Hrbas and Tomislav Barth
    Cross-reactivity of anti-oxytocin sera
    1982, Vol. 47, Issue 6, pp. 1654–1658 [Abstract]
  • Michal Lebl, Jan Pospíšek, Jan Hlaváček, Tomislav Barth, Petr Maloň, Linda Servítová, Karel Hauzer and Karel Jošt
    Analogues of neurohypophysial hormones, containing tert-leucine: Synthesis and properties
    1982, Vol. 47, Issue 2, pp. 689–701 [Abstract]
  • Zdenko Procházka, Jorga Smolíková, Petr Maloň and Karel Jošt
    Synthetic utilization of α-amino-γ-bromobutyric acid in the preparation of non-coded amino acids; IR study of homoserine
    1981, Vol. 46, Issue 11, pp. 2935–2946 [Abstract]
  • Tomislav Barth, Jiřina Slaninová, Linda Servítová, Michal Lebl, Christine Kotsira-Engonopoulos, Chrysa Tzougraki, Iphigenia Photaki, Milan Krojidlo and Karel Jošt
    The effect of some structural modifications of the oxytocin molecule on the duration of the galactogogic response
    1981, Vol. 46, Issue 10, pp. 2441–2445 [Abstract]
  • Jana Škopková, Pavel Hrbas, Jiřina Slaninová and Tomislav Barth
    Prolonged antidiuretic action of vasopressin analogues in relation to their primary structure
    1981, Vol. 46, Issue 8, pp. 1850–1855 [Abstract]
  • Jiřina Slaninová, Michal Lebl, Tomislav Barth and Karel Jošt
    The effect of magnesium ions on the uterotonic activity of carba analogues of oxytocin modified in position 4
    1981, Vol. 46, Issue 7, pp. 1689–1692 [Abstract]
  • Zdenko Procházka, Michal Lebl, Linda Servítová, Tomislav Barth and Karel Jošt
    Synthesis and pharmacological properties of [2-p-fluorophenylalanine]deamino-1-carba-oxytocin and its diastereoisomeric sulfoxides
    1981, Vol. 46, Issue 4, pp. 947–956 [Abstract]
  • Asja Šiševa, Ljuben M. Sirakov, Jiřina Slaninová and Tomislav Barth
    Biological activity of some insulin derivatives
    1981, Vol. 46, Issue 1, pp. 300–302 [Abstract]
  • Pavel Hrbas, Jiřina Slaninová, Tomislav Barth and František Franěk
    Cross-reactivity study of oxytocin antibodies with oxytocin and its analogues modified in the cyclic part of the molecule
    1981, Vol. 46, Issue 1, pp. 270–277 [Abstract]
  • Tomislav Barth, Jiřina Slaninová, Michal Lebl and Karel Jošt
    Biological activities and protracted action of carba-analogues of deamino-oxytocin with O-methyltyrosine in position 2
    1980, Vol. 45, Issue 11, pp. 3045–3050 [Abstract]
  • Michal Lebl
    High-performance liquid chromatography of carba-analogues of oxytocin; a method for the determination of sulfides and sulfoxides in peptides
    1980, Vol. 45, Issue 11, pp. 2927–2937 [Abstract]
  • Michal Lebl, Tomislav Barth, Jana Škopková and Karel Jošt
    Synthesis and some pharmacological properties of [7-glycine, 8-ornithine]vasopressin and two of its analogues
    1980, Vol. 45, Issue 10, pp. 2865–2871 [Abstract]
  • Michal Lebl, Tomislav Barth and Karel Jošt
    Synthesis and pharmacological properties of oxytocin analogues modified simultaneously in position 2 and in the disulfide bridge
    1980, Vol. 45, Issue 10, pp. 2855–2864 [Abstract]
  • Michal Lebl, Alena Machová, Pavel Hrbas, Tomislav Barth and Karel Jošt
    Analogues of deamino-1-carba-oxytocin with an aliphatic amino acid in position 4: chemical synthesis and biological activities
    1980, Vol. 45, Issue 10, pp. 2714–2723 [Abstract]
  • Zdenko Procházka and Karel Jošt
    L-Cystathionine derivatives for the synthesis of peptides
    1980, Vol. 45, Issue 7, pp. 1982–1990 [Abstract]
  • Zdenko Procházka and Karel Jošt
    Synthesis of the amino-terminal decapeptide of human calcitonin, in which the disulfide bond is replaced by a thioether group
    1980, Vol. 45, Issue 4, pp. 1305–1314 [Abstract]
  • Michal Lebl, Vera Bojanovska, Tomislav Barth and Karel Jošt
    Synthesis and properties of oxytocin analogues acting as irreversible inhibitors of the uterotonic response to oxytocin
    1979, Vol. 44, Issue 8, pp. 2573–2582 [Abstract]
  • Michal Lebl, Tomislav Barth and Karel Jošt
    Analogues of oxytocin with esters of glutamic acid instead of glutamine in position 4: Synthesis of a compound with high and specific galactogogic activity
    1979, Vol. 44, Issue 8, pp. 2563–2572 [Abstract]
  • Michal Lebl, Anastasia Dimeli, Vera Bojanovska, Jiřina Slaninová, Tomislav Barth and Karel Jošt
    Synthesis and some biological properties of amides derived from [4-glutamic acid]deamino-1-carba-oxytocin
    1979, Vol. 44, Issue 8, pp. 2556–2562 [Abstract]
  • Asja Šiševa, Jiřina Slaninová, Tomislav Barth, Stephan P. Ditzov and Luben M. Sirakov
    Isoelectric focusing of insulin, 125I-insulin and the 125I-insulin-antibody complex
    1979, Vol. 44, Issue 6, pp. 1828–1834 [Abstract]
  • Tomislav Barth, Asja Šiševa, Ljuben Sirakov, Jiřina Slaninová and Stefan Ditzov
    Cross-reaction of some insulin derivatives with anti-insulin serum
    1978, Vol. 43, Issue 11, pp. 2967–2972 [Abstract]
  • Michal Lebl, Tomislav Barth and Karel Jošt
    Synthesis, reduction, and pharmacological properties of the sulfoxides of some carba-analogues of oxytocin
    1978, Vol. 43, Issue 6, pp. 1538–1556 [Abstract]
  • Michal Lebl, Tomislav Barth and Karel Jošt
    Nα-Glycyl-glycyl-glycyl-8-ornithine-vasopressin: A trypsin resistant vasopressin analog with a specific pressor effect
    1978, Vol. 43, Issue 5, pp. 1300–1305 [Abstract]
  • Zdenko Procházka, Ivan Krejčí, Běla Kupková, Jiřina Slaninová, Vera Bojanovska, Zdeněk Prusík, Ilse A. Vosekalna, Petr Maloň, Tomislav Barth, Ivo Frič, Karel Bláha and Karel Jošt
    Synthesis and properties of the Nα-glycyl-glycyl-glycyl-8-lysine-vasopressin and its des-glycinamide derivative
    1978, Vol. 43, Issue 5, pp. 1285–1299 [Abstract]
  • Jiřina Slaninová, Tomislav Barth, Jana Škopková, Ivo Bláha and František Franěk
    Preparation of antibodies to [8-D-arginine]deamino-vasopressin and study of their cross-reactivity with vasopressin analogues
    1978, Vol. 43, Issue 4, pp. 1167–1174 [Abstract]
  • Zdenko Procházka, Tomislav Barth, Joseph H. Cort, Karel Jošt and František Šorm
    Synthesis and some pharmacological properties of [8-L-arginine]deamino-1-carba-vasopressin
    1978, Vol. 43, Issue 2, pp. 655–663 [Abstract]
  • Michal Lebl and Karel Jošt
    Synthesis of [4-glutamic acid]deamino-1-carba-oxytocin
    1978, Vol. 43, Issue 2, pp. 523–534 [Abstract]