Collect. Czech. Chem. Commun. 2003, 68, 1275-1294

On the Relationship between the Structure and Antimycobacterial Activity of Substituted N-Benzylsalicylamides

Karel Waissera,*, Milan Peřinaa, Věra Klimešováa and Jarmila Kaustováb

a Department of Inorganic and Organic Chemistry, Faculty of Pharmacy, Heyrovského 1203, CZ-500 05 Hradec Králové, Czech Republic
b National Reference Laboratory for Mycobacterium kansasii, Institute of Hygiene, Partyzánské nám. 7, CZ-728 92 Ostrava, Czech Republic

Individual author index pages

Other CCCC articles of these authors

  • Karel Waisser*, Miloš Macháček, Hynek Dostál, Jiří Gregor, Lenka Kubicová, Věra Klimešová, Jiří Kuneš, Karel Palát, Jr., Jana Hladůvková, Jarmila Kaustová and Ute Möllmann
    Relationships Between the Chemical Structure of Substances and Their Antimycobacterial Activity Against Atypical Strains. Part 18. 3-Phenyl-2H-1,3-benzoxazine-2,4(3H)-diones and Isosteric 3-Phenylquinazoline-2,4(1H,3H)-diones
    1999, Vol. 64, Issue 11, pp. 1902–1924 [Abstract]
  • Miroslav Holík*, Zdeněk Friedl, Karel Waisser and Jiří Gregor
    Multivariate Regression with Substituent Shift Increments. IV. 2-(4-X-Phenyl)-1,3-dihydro-2H-isoindole-1,3-diones and 3-(4-X-Phenyl)-3,4-dihydro-2H-1,3-benzoxazine-2,4-diones
    1999, Vol. 64, Issue 10, pp. 1709–1726 [Abstract]
  • Karel Waisser*, Karel Palát, Jr. and Otto Exner*
    Substituent Effects on Conformational Equilibria: Substituted Thiobenzanilides
    1999, Vol. 64, Issue 8, pp. 1295–1306 [Abstract]
  • Věra Klimešová*, Martin Svoboda, Karel Waisser, Milan Pour and Jarmila Kaustová
    Synthesis and Antimicrobial Activity of New 4-(Benzylsulfanyl)pyridine Derivatives
    1999, Vol. 64, Issue 2, pp. 417–434 [Abstract]
  • Jiří Kuneš, Jiří Jáchym, Petr Jirásko, Želmíra Odlerová and Karel Waisser
    Combination of the Topliss Approach with the Free-Wilson Analysis in the Study of Antimycobacterial Activityof 4-Alkylthiobenzanilides
    1997, Vol. 62, Issue 9, pp. 1503–1510 [Abstract]
  • Katarína Kráľová, František Šeršeň, Věra Klimešová and Karel Waisser
    Effect of 2-Alkylthio-4-pyridinecarbothiamides on Photosynthetic Electron Transport in Spinach Chloroplasts
    1997, Vol. 62, Issue 3, pp. 516–520 [Abstract]
  • Hans-Dietrich Stachel, Želmíra Odlerová and Karel Waisser
    A New Pharmacophore of Potential Antimycobacterial Activity: The Disulfide Group in the Ring of Alicyclic Compounds
    1997, Vol. 62, Issue 3, pp. 510–515 [Abstract]
  • Karel Waisser, Jiří Kuneš, Alexandr Hrabálek, Miloš Macháček and Želmíra Odlerová
    New Groups of Potential Antituberculotics: 5-Alkylthio-1-aryltetrazoles
    1996, Vol. 61, Issue 5, pp. 791–798 [Abstract]
  • Karel Waisser, Jiří Kuneš, Alexandr Hrabálek and Želmíra Odlerová
    New Groups of Potential Antituberculotics: Bis(1-aryltetrazol-5-yl) Disulfides. Structure Activity Relationship
    1994, Vol. 59, Issue 1, pp. 234–238 [Abstract]
  • Karel Waisser, Lenka Kubicová, Věra Klimešová and Želmíra Odlerová
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    1993, Vol. 58, Issue 12, pp. 2977–2982 [Abstract]
  • Věra Klimešová
    Preparation of Some Thio Derivatives of Pyridinecarbothioamides
    1993, Vol. 58, Issue 5, pp. 1195–1197 [Abstract]
  • Karel Waisser, Lenka Kubicová and Želmíra Odlerová
    Antituberculotic 4'-Cyclohexylthiobenzanilides: Combination of Free-Wilson Method in QSAR with Topliss Approach
    1993, Vol. 58, Issue 1, pp. 205–212 [Abstract]
  • Karel Waisser, Miloš Macháček, Želmíra Odlerová, Wilfried Thiel and Roland Mayer
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    1993, Vol. 58, Issue 1, pp. 197–204 [Abstract]
  • Karel Waisser, Jiří Kuneš, Jiří Klimeš, Miroslav Polášek and Želmíra Odlerová
    Relations between Structure and Antituberculotic Activity of 4-Alkoxybenzoic Acids
    1993, Vol. 58, Issue 1, pp. 191–196 [Abstract]
  • Karel Waisser, Jiří Kuneš and Želmíra Odlerová
    Correlation of structural parameters with antituberculotic activity in a group of 2-benzamidobenzothiazoles
    1991, Vol. 56, Issue 12, pp. 2978–2985 [Abstract]
  • Miroslav Polášek, Karel Waisser and Tomáš Bouček
    Determination of the substituent constant σp- for the thioamide group -CSNH2 from the ionization of anilines and phenols
    1991, Vol. 56, Issue 12, pp. 2964–2968 [Abstract]
  • Karel Waisser and Jana Bořková
    Relations between structure and antituberculotic activity in a group of 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
    1991, Vol. 56, Issue 11, pp. 2395–2401 [Abstract]
  • Karel Waisser, Jiří Vanžura, Alexandr Hrabálek, Jarmila Vinšová, Štefan Grešák, Jiří Hruška and Želimíra Odlerová
    Antimycobacterial derivatives of tetrazole
    1991, Vol. 56, Issue 11, pp. 2389–2394 [Abstract]
  • Karel Waisser, Nestor Houngbedji, Miloš Macháček, Miroslav Sekera, Josef Urban and Želmíra Odlerová
    Antimycobacterial thiobenzanilides
    1990, Vol. 55, Issue 1, pp. 307–316 [Abstract]
  • Naďa Zimová, Ivan Němec, Miroslava Ehlová and Karel Waisser
    The effect of the structure of the substituent in position ten on the voltammetric behaviour of phenothiazin derivatives
    1990, Vol. 55, Issue 1, pp. 63–71 [Abstract]
  • Karel Waisser, Miloš Macháček, Jean Lebvoua, Jiří Hrbata and Jaroslav Dršata
    Quantitative relations between chemical structure and hepatotoxicity of thiobenzamides
    1988, Vol. 53, Issue 11, pp. 2957–2961 [Abstract]
  • Otto Exner and Karel Waisser
    Dipole moment and electron distribution of the thioamide group
    1982, Vol. 47, Issue 3, pp. 828–837 [Abstract]