Collect. Czech. Chem. Commun. 1993, 58, 893-901
https://doi.org/10.1135/cccc19930893

New Preparation of 2-N-Alkyl(aryl)amino-5-methyl-4H-1,3-thiazin-4-ones and 3,4-Dihydro-5-methyl-2,4-dioxo-2H-1,3-thiazine

Dušan Koščík, Milan Dzurilla and Peter Kutschy

Department of Organic Chemistry, Šafárik University,041 67 Košice, Slovak Republic

Individual author index pages


Other CCCC articles of these authors

  • Peter Kutschy*, Andrej Sýkora, Zuzana Čurillová, Mária Repovská, Martina Pilátová, Ján Mojžiš, Roman Mezencev, Pavel Pazdera and Tatiana Hromjáková
    Glyoxyl analogs of indole phytoalexins: Synthesis and anticancer activity
    2010, Vol. 75, Issue 8, pp. 887–903 [Abstract]
  • Martin Humeník*, Peter Kutschy, Vladimír Kováčik and Slávka Bekešová
    1,2-Anhydrosaccharides and 1,2-Cyclic Sulfites as Saccharide Donors in Convergent Synthesis of Glucopyranosyl-, Mannopyranosyl- and Ribofuranosylbenzocamalexin
    2005, Vol. 70, Issue 4, pp. 487–506 [Abstract]
  • Martin Humeník*, Peter Kutschy, Katarína Valková, Branislav Horváth, Vladimír Kováčik and Slávka Bekešová
    Synthesis of β-D-Glucopyranosides of 6-Substituted 2-(Indol-3-yl)benzothiazoles
    2005, Vol. 70, Issue 1, pp. 72–84 [Abstract]
  • Martin Humeník*, Milan Dzurilla, Peter Kutschy, Eva Solčániová, Vladimír Kováčik and Slávka Bekešová
    Synthesis of 1-Glycosyl Derivatives of Benzocamalexin
    2004, Vol. 69, Issue 8, pp. 1657–1674 [Abstract]
  • Peter Kutschy*, Marian Sabol, Renata Marušková, Zuzana Čurillová, Milan Dzurilla, Imrich Géci, Juraj Alföldi and Vladimír Kováčik
    A Linear Synthesis of 1-(β-D-Glucopyranosyl)brassinin, -brassenin A, -brassenin B and 9-(β-D-Glucopyranosyl)cyclobrassinin
    2004, Vol. 69, Issue 4, pp. 850–866 [Abstract]
  • Janka Záletová, Milan Dzurilla, Peter Kutschy*, Pavel Pazdera, Vladimír Kováčik, Juraj Aldölfi and Slávka Bekešová
    Synthesis of 4,6-Disubstituted-2-(1H-indol-3-yl)benzothiazoles
    2004, Vol. 69, Issue 2, pp. 453–460 [Abstract]
  • Peter Kutschy*, Mojmír Suchý, Milan Dzurilla, Mitsuo Takasugi and Vladimír Kováčik
    A New Approach to Imidazo[1,5-a]indole Derivatives
    2000, Vol. 65, Issue 7, pp. 1163–1172 [Abstract]
  • Peter Kutschy*, Mojmír Suchý, Milan Dzurilla, Pavel Pazdera, Mitsuo Takasugi and Vladimír Kováčik
    Spirocyclization of Isatin with Chiral α-Aminothiols: Diastereoselective Synthesis of (-)- and (+)-4'-(Methoxycarbonyl)spiro[indoline-3,2'-thiazolidin]-2-one
    2000, Vol. 65, Issue 3, pp. 425–433 [Abstract]
  • Milan Dzurilla*, Martin Ružinský, Peter Kutschy, Jalpa P. Tewari and Vladimír Kováčik
    Application of 2-Substituted Ethyl Isothiocyanates and 2-Aminothiols in the Synthesis of the Analogs of Indole Phytoalexin Camalexin
    1999, Vol. 64, Issue 9, pp. 1448–1456 [Abstract]
  • Peter Kutschy*, Milan Dzurilla, Mitsuo Takasugi and Adriana Sabová
    Synthesis of Some Analogs of Indole Phytoalexins Brassinin and Methoxybrassenin B and Their Positional Isomers
    1999, Vol. 64, Issue 2, pp. 348–362 [Abstract]
  • Milan Dzurilla, Peter Kutschy, Jalpa P. Tewari, Martin Ružinský, Stanislav Šenvický and Vladimír Kováčik
    Synthesis and Antifungal Activity of New Indolylthiazinone Derivatives
    1998, Vol. 63, Issue 1, pp. 94–102 [Abstract]
  • Oľga Hritzová, Gejza Suchár, Ivan Danihel and Peter Kutschy
    Solvent Effect on the Structure and Infrared Spectra of N-(3-Chloro-2-benzo[b]thienocarbonyl)-N'-ethylthiourea
    1996, Vol. 61, Issue 11, pp. 1620–1626 [Abstract]
  • Milan Dzurilla, Peter Kutschy, Ján Imrich and Stanislav Brtoš
    Hugershoff Reaction of N-1- or N-2-Naphthoyl-N'-monosubstituted and N',N'-Disubstituted Thiourea Derivatives
    1994, Vol. 59, Issue 12, pp. 2663–2676 [Abstract]
  • Vlastimír Ficeri, Peter Kutschy, Milan Dzurilla and Ján Imrich
    [3,3]- Versus [1,3]-Sigmatropic Rearrangement of O-Substituted Allyl N-Acylmonothiocarbamates
    1994, Vol. 59, Issue 12, pp. 2650–2662 [Abstract]
  • Marcel Török, Milan Dzurilla, Peter Kutschy, Ján Imrich, Ivan Danihel, Paul Rademacher and Heinz Bandmann
    Cyclohexylideneacetyl Isothiocyanate. Precursor for the Synthesis of 1,3-Thiazaspirocycloalkanes and 1,3-Diazaspirocycloalkanes
    1994, Vol. 59, Issue 5, pp. 1203–1210 [Abstract]
  • Oľga Hritzová and Dušan Koščík
    Intramolecular Hydrogen Bonds and Fermi Resonance in N-Substituted N'-(2-Fluorobenzoyl)thiourea Derivatives
    1994, Vol. 59, Issue 4, pp. 951–956 [Abstract]
  • Peter Kutschy, Milan Dzurilla, Vlastimír Ficeri and Dušan Koščík
    New Synthesis of N-Acylurea Derivatives
    1993, Vol. 58, Issue 3, pp. 575–587 [Abstract]
  • Milan Dzurila, Peter Kutschy, Ján Imrich, Dušan Koščík and Robert Kraus
    Cyclization and oxidation of N-substituted phenyl-N’-(2-methyl-3-phenylpropenoyl)thioureas
    1991, Vol. 56, Issue 6, pp. 1287–1294 [Abstract]
  • Oľga Hritzová and Dušan Koščík
    Hydrogen bonds in derivatives of N-substituted N’-benzoyl- and N’-(2-chlorobenzoyl)thiourea
    1991, Vol. 56, Issue 4, pp. 880–885 [Abstract]
  • Milan Dzurilla, Peter Kutschy, Dušan Koščík and Štefan Toma
    Intramolecular cyclization of O-alkyl-N-(3-phenylpropenoyl)thiocarbamates catalyzed by boron trifluoride
    1990, Vol. 55, Issue 3, pp. 710–717 [Abstract]
  • Oľga Hritzová, Peter Kutschy, Ján Imrich and Thomas Schöffmann
    Hydrogen bonds in N-(3-chloro-2-benzo[b]thienocarbonyl)- and N-(2-benzo[b]thienocarbonyl)-N'-monosubstituted thioureas
    1987, Vol. 52, Issue 11, pp. 2673–2679 [Abstract]
  • Milan Dzurilla, Peter Kutschy and Dušan Koščík
    A new method for preparation of 1-(4-substituted phenyl)-6-phenyl-2-thiouracils via cyclization of N-(4-substituted phenyl)-N'-3-phenylpropenoylthioureas and Dimroth rearrangement of 2-(4-substituted phenylimino)-6-phenyl-5,6-dihydro-4H-1,3-thiazin-4-ones
    1987, Vol. 52, Issue 9, pp. 2260–2265 [Abstract]
  • Peter Kutschy, Milan Dzurilla, Dušan Koščík and Pavol Kristian
    An advantageous synthesis of S-(2-propenyl) N-acylmonothiocarbamates by [3,3]-sigmatropic rearrangement of O-(2-propenyl) N-acylmonothiocarbamates
    1987, Vol. 52, Issue 7, pp. 1764–1772 [Abstract]
  • Peter Kutschy, Pavol Kristian, Milan Dzurilla, Dušan Koščík and Róbert Nádaskay
    Selectivity of nucleophilic addition to and substitution at isothiocyanatocarbonyl group. Reactions of 4-pentinoyl- and 2-(2-propinyl)-4-pentinoyl isothiocyanate with amines and methanol
    1987, Vol. 52, Issue 4, pp. 995–1005 [Abstract]
  • Milan Dzurilla, Ondrej Forgáč, Peter Kutschy, Pavol Kristian, Dušan Koščík and Ján Imrich
    Synthesis of 1,3-diazaspiro[5,5]undecanes and 1-thia-3-azaspiro[5,5]undec-2-enes by reaction of 2-cyanocyclohexylideneacetyl isothiocyanate with amines and sodium hydrogen sulfide
    1987, Vol. 52, Issue 4, pp. 989–994 [Abstract]
  • Peter Kutschy, Ján Imrich, Juraj Bernát, Pavol Kristian, Oľga Hritzová and Thomas Schöffmann
    Photocyclization of N-(3-chloro-2-benzo[b]thienocarbonyl)-N'-monosubstituted thioureas
    1986, Vol. 51, Issue 12, pp. 2839–2847 [Abstract]
  • Peter Kutschy, Ján Imrich, Juraj Bernát, Pavol Kristian and Iveta Fedoriková
    A study of photocyclization of O-alkyl N-(3-chloro-2-benzo[b]thienocarbonyl)monothiocarbamates
    1986, Vol. 51, Issue 9, pp. 2002–2012 [Abstract]
  • Peter Kutschy, Milan Dzurilla, Ladislav Kniežo, Juraj Bernát, Ján Imrich, Pavol Kristian and Róbert Nádaskay
    Reactions of 3-butine-2-methyl-2-ol with isothiocyanates
    1986, Vol. 51, Issue 5, pp. 1119–1126 [Abstract]
  • Gejza Suchár, Milan Dzurilla and Pavol Kristian
    A study of dipole moments of substituted isothiocyanates of 1,3-diphenyl-2-propen-1-one
    1984, Vol. 49, Issue 10, pp. 2382–2386 [Abstract]
  • Pavol Kristian, Dušan Koščík and Jozef Gonda
    Heterocycles with a pyrido[3,2-e]-1,3-selenazine and pyrido[3,4-e]-1,3-selenazine ring systems
    1983, Vol. 48, Issue 12, pp. 3567–3574 [Abstract]
  • Dušan Koščík, Pavol Kristian and Ondrej Forgáč
    Synthesis of 2-amino-5,7-dimethyl-4-oxopyrido[3,4-e]-1,3-thiazines
    1983, Vol. 48, Issue 12, pp. 3426–3432 [Abstract]
  • Dušan Koščík, Pavol Kristian, Jozef Gonda and Emília Dandárová
    New synthesis of 2-amino-4-oxopyrido[3,2-e]-1,3-thiazines and 1-alkyl(aryl)pyrido[3,2-e]-2-thiouracils
    1983, Vol. 48, Issue 11, pp. 3315–3328 [Abstract]
  • Milan Dzurilla, Pavol Kristian, Ján Imrich and Juraj Štec
    Bromine oxidation of N-(3 or 4-substituted phenyl)-N'-3-phenylpropenoylthioureas
    1983, Vol. 48, Issue 11, pp. 3134–3139 [Abstract]
  • Peter Kutschy, Pavol Kristian, Miloslava Dandárová and Jaroslav Kováč
    Synthesis and reactions of cis-3-(2-furyl)propenoyl isocyanate
    1981, Vol. 46, Issue 5, pp. 1160–1166 [Abstract]
  • Peter Kutschy, Milan Dzurilla, Pavol Kristian and Kvetoslava Kutschyová
    Synthesis of 2-substituted 5-arylidenethiazolin-4-ones from α,β-unsaturated acyl isothiocyanates
    1981, Vol. 46, Issue 2, pp. 436–445 [Abstract]
  • Milan Dzurilla, Pavol Kristian and Peter Kutschy
    Synthesis of 2-amino-6-substituted 5,6-dihydro-4H-1,3-thiazin-4-ones from α,β-unsaturated acyl isothiocyanates
    1980, Vol. 45, Issue 11, pp. 2958–2964 [Abstract]
  • Ján Imrich, Pavol Kristian, Dušan Podhradský and Milan Dzurilla
    Kinetics of reactions of acyl isothiocyanates with amines
    1980, Vol. 45, Issue 8, pp. 2334–2342 [Abstract]
  • Peter Kutschy, Pavol Kristian, Milan Dzurilla and Jaroslav Kováč
    Reactions of α,β-unsaturated acyl isothiocyanates with phenylhydrazine
    1980, Vol. 45, Issue 6, pp. 1692–1703 [Abstract]
  • Pavol Kristian, Peter Kutschy and Milan Dzurilla
    Synthesis of 2,2,4-trisubstituted 2H-1,3-oxazetes from acyl isothiocyanates
    1979, Vol. 44, Issue 4, pp. 1324–1333 [Abstract]