Collect. Czech. Chem. Commun. 1965, 30, 3730-3743
https://doi.org/10.1135/cccc19653730

5-Arylpyrimidine II. 4,6-Disubstituierte 5-Phenylpyrimidine

Z. Buděšínský, F. Roubínek and E. Svátek

Individual author index pages


Other CCCC articles of these authors

  • Z. Buděšínský, P. Lederer and J. Daněk
    3-(3-Amino-2-hydroxypropyl)- and 3-(3-aminoacetonyl)-4(3H)-quinazolines
    1977, Vol. 42, Issue 12, pp. 3473–3486 [Abstract]
  • V. Vosátka, A. Čapek and Z. Buděšínský
    O-(2-Methylthio-5-pyrimidinyl) thiocarbamates and their antimycotic activity
    1977, Vol. 42, Issue 11, pp. 3186–3191 [Abstract]
  • M. Rajšner, E. Svátek, J. Metyšová, M. Bartošová, F. Mikšík and M. Protiva
    Fluorinated tricyclic neuroleptics with prolonged effects: Some new 8-chloro-3-fluoro-10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
    1977, Vol. 42, Issue 10, pp. 3079–3093 [Abstract]
  • I. Červená, K. Šindelář, Z. Kopicová, J. Holubek, E. Svátek, J. Metyšová, M. Hrubantová and M. Protiva
    Fluorinated tricyclic neuroleptics: 6,7-Difluoro derivative of chlorprothixene and 2-fluoro-3-hydroxy derivative of octoclothepin
    1977, Vol. 42, Issue 6, pp. 2001–2017 [Abstract]
  • I. Červená, K. Šindelář, J. Metyšová, E. Svátek, M. Ryska, M. Hrubantová and M. Protiva
    New potential neuroleptics of the perathiepin and octoclothepin series: 8-Chloro-7-methoxy, 8-chloro-7-trifluoromethyl- and 7-fluoro-8-methyl-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1977, Vol. 42, Issue 5, pp. 1705–1722 [Abstract]
  • Z. J. Vejdělek, B. Kakáč, J. Holubek, E. Svátek, M. Bartošová and M. Protiva
    1,2,3,4,7,8-Hexahydro-6H-cyclopent[g]isoquinoline and N-substituted derivatives; Synthesis and pharmacological screening
    1977, Vol. 42, Issue 4, pp. 1200–1208 [Abstract]
  • J. Sluka, J. Novák and Z. Buděšínský
    2-Phenylbenzimidazoles as potential anthelminthics
    1976, Vol. 41, Issue 12, pp. 3628–3634 [Abstract]
  • R. Smrž, J. O. Jílek, B. Kakáč, J. Holubek, E. Svátek, M. Bartošová and M. Protiva
    2(8)-Chloro-10(11)-(dimethylaminoalkyl)dibenzo[b,f]thiepins as potential CNS agents; Synthesis and pharmacological screening
    1976, Vol. 41, Issue 11, pp. 3420–3436 [Abstract]
  • Z. Buděšínský, P. Lederer, F. Roubínek, A. Šváb and J. Vavřina
    Alkoxy-2,4-quinazolinediamines
    1976, Vol. 41, Issue 11, pp. 3405–3414 [Abstract]
  • J. Sluka, J. Novák and Z. Buděšínský
    Ethers of 5-halogenosalicylic and thiosalicylic acids
    1976, Vol. 41, Issue 11, pp. 3384–3390 [Abstract]
  • R. Smrž, J. O. Jílek, K. Šindelář, B. Kakáč, E. Svátek, J. Holubek, J. Grimová and M. Protiva
    5(or 4)-Arylthio-2-methylthiopyrimidines as potential intermediates in the synthesis of tricyclic pyrimido systems
    1976, Vol. 41, Issue 9, pp. 2771–2787 [Abstract]
  • K. Šindelář, B. Kakáč, J. Holubek, E. Svátek, M. Ryska, J. Metyšová and M. Protiva
    Potential metabolites of neuroleptics of the 10-piperazino-10,11-dihydrodibenzo[b,f]thiepin series: 2,3-Dihydroxy derivatives of perathiepin and octoclothepin and some related compounds
    1976, Vol. 41, Issue 5, pp. 1396–1415 [Abstract]
  • K. Šindelář, J. O. Jílek, V. Bártl, J. Metyšová, B. Kakáč, J. Holubek, E. Svátek, J. Pomykáček and M. Protiva
    Neuroleptics of the 10-piperazino-10,11-dihydrodibenzo[b,f]thiepin series and related substances: Piperazine-alkylated homologues of octoclothepin and methiothepin, 5,5-dimethyl-10,11-dihydro-5H-dibenzo[b,f]silepin analogue of perathiepin
    1976, Vol. 41, Issue 3, pp. 910–922 [Abstract]
  • I. Červená, J. Metyšová, E. Svátek, B. Kakáč, J. Holubek, M. Hrubantová and M. Protiva
    Potent neuroleptics with prolonged activity and diminished toxicity: 7,8-Dihalogeno-10-piperazinodibenzo[b,f]thiepins
    1976, Vol. 41, Issue 3, pp. 881–905 [Abstract]
  • J. O. Jílek, I. Červená, Z. Kopicová, K. Šindelář, E. Svátek, J. Metyšová, A. Dlabač, J. Pomykáček and M. Protiva
    Potent neuroleptic agents: Some new amino alcohols of the 10-piperazinodibenzo[b,f]thiepin series and their derivatives
    1976, Vol. 41, Issue 2, pp. 443–458 [Abstract]
  • K. Šindelář, A. Dlabač, B. Kakáč, E. Svátek, J. Holubek, Z. Šedivý, E. Princová and M. Protiva
    Noncataleptic potential neuroleptics: 2-Acetamido-, 2-amino- and 2-acetyl derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1975, Vol. 40, Issue 9, pp. 2649–2666 [Abstract]
  • Z. Kopicová, E. Svátek and M. Protiva
    Potential tetracyclic neuroleptics: 12-(4-Methylpiperazino)benzo[b]naphtho[2,3-f]thiepin and its 12,13-dihydro derivative
    1975, Vol. 40, Issue 6, pp. 1960–1965 [Abstract]
  • K. Šindelář, A. Dlabač, J. Metyšová, B. Kakáč, J. Holubek, E. Svátek, Z. Šedivý and M. Protiva
    Potential antipsychotics: 2-Methoxy, 2-methylthio-, 2-(dimethylsulfamoyl)- and 2-trifluoromethyl-10-piperazinodibenzo[b,f]thiepins
    1975, Vol. 40, Issue 6, pp. 1940–1959 [Abstract]
  • M. Rajšner, E. Svátek, J. Metyšová and M. Protiva
    12-(3-dimethylaminopropylidene)-12H-benzo[f]naphtho[1,8-bc]thiepin and 10-chloro-12-(4-methylpiperazino)-12H-benzo[f]naphtho[1,8-bc]thiepin
    1975, Vol. 40, Issue 5, pp. 1604–1611 [Abstract]
  • Z. Buděšínský, J. Sluka, J. Novák and J. Daněk
    5-Styryl-2-benzimidazolylurethanes as potential anthelminthics
    1975, Vol. 40, Issue 4, pp. 1089–1094 [Abstract]
  • Z. Buděšínský, L. Brůna, A. Šváb and A. Čapek
    5-(3-Iodopropargyloxy)pyrimidines as effective fungistatics
    1975, Vol. 40, Issue 4, pp. 1078–1088 [Abstract]
  • M. Rajšner, J. Metyšová, E. Svátek, F. Mikšík and M. Protiva
    2- And 3-fluoro derivatives of clorotepin and related compounds; 6- And 7-fluoro derivative of chlorprothixene
    1975, Vol. 40, Issue 3, pp. 719–737 [Abstract]
  • I. Červená, E. Svátek, J. Metyšová and M. Protiva
    11-Piperazino-8,9-dihydro(and 8,9,11,12-tetrahydro)-7H-benz[b]indeno[5,6-f]thiepins
    1974, Vol. 39, Issue 12, pp. 3733–3740 [Abstract]
  • K. Šindelář, J. Metyšová, B. Kakáč, J. Holubek, E. Svátek, J. O. Jílek, J. Pomykáček and M. Protiva
    8-Acyl derivatives of 10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1974, Vol. 39, Issue 8, pp. 2099–2114 [Abstract]
  • M. Rajšner, E. Svátek, J. Metyš and M. Protiva
    Geometric isomerism of 4-(3-dimethylaminopropylidene)-9H-thieno[2,3-b]benzo[e]thiepin
    1974, Vol. 39, Issue 5, pp. 1366–1376 [Abstract]
  • K. Šindelář, B. Kakáč, E. Svátek, J. Holubek, M. Rajšner, J. Metyšová and M. Protiva
    9-Chloro-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin and some related synthetic experiments
    1974, Vol. 39, Issue 1, pp. 333–354 [Abstract]
  • K. Šindelář, M. Rajšner, I. Červená, V. Valenta, J. O. Jílek, K. Kakáč, J. Holubek, E. Svátek, F. Mikšík and M. Protiva
    Neurotropic and psychotropic agents. LXVII. 1-[4,4-Bis(4-fluorophenyl)butyl]-4-hydroxy-4-(3-trifluoromethyl-4-chlorophenyl)piperidine and related compounds: New synthetic approaches
    1973, Vol. 38, Issue 12, pp. 3879–3901 [Abstract]
  • K. Šindelář, B. Kakáč, E. Svátek, J. Holubek, J. Metyšová, M. Hrubantová and M. Protiva
    Neurotropic and psychotropic agents. LXVI. 6,8-Dichloro- and 6,9-dichloro-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin
    1973, Vol. 38, Issue 11, pp. 3321–3338 [Abstract]
  • V. Bártl, E. Svátek and M. Protiva
    Neurotropic and psychotropic agents. LIX. 3-Methoxy-11-(3-dimethylaminopropylidene)-6H,11H-dibenzo[b,e]thiepin and some related compounds
    1973, Vol. 38, Issue 5, pp. 1596–1601 [Abstract]
  • K. Šindelář, B. Kakáč, E. Svátek, J. Metyšová and M. Protiva
    Neurotropic and psychotropic agents. LVIII. 8-Hydroxy-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin, O-substitution derivatives and some related compounds
    1973, Vol. 38, Issue 5, pp. 1579–1595 [Abstract]
  • J. O. Jílek, J. Metyšová, E. Svátek, F. Jančik, J. Pomykáček and M. Protiva
    Neurotropic and psychotropic agents. LVI. Sulfoxides, N-oxides and sulfones derived from neuroleptic 10-piperazino-10,11-dihydrodibenzo[b,f]thiepins
    1973, Vol. 38, Issue 2, pp. 599–610 [Abstract]
  • J. O. Jílek, K. Šindelář, J. Pomykáček, O. Horešovský, K. Pelz, E. Svátek, B. Kakáč, J. Holubek, J. Metyšová and M. Protiva
    Neurotropic and psychotropic compounds. LV. New syntheses of 8-chloro-10-(4-methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin and related compounds
    1973, Vol. 38, Issue 1, pp. 115–131 [Abstract]
  • F. Kvis, E. Svátek, R. Zahradník and M. Protiva
    Benzocycloheptenes and heterocyclic analogues as potential drugs. VII. 4-Phenyl-2,3,4,5-tetrahydro-1-benzothiepins and some related compounds
    1972, Vol. 37, Issue 11, pp. 3808–3816 [Abstract]
  • K. Šindelář, E. Svátek and M. Protiva
    Neurotropic and psychotropic compounds. LIV. 2-(2-Thienylselenomethyl)benzoic acid and its transformations
    1972, Vol. 37, Issue 11, pp. 3660–3663 [Abstract]
  • Z. Buděšínský and P. Lederer
    A new synthesis of the quinazoline nucleus
    1972, Vol. 37, Issue 8, pp. 2779–2785 [Abstract]
  • M. Protiva, V. Seidlová, E. Svátek, B. Kakáč and J. Holubek
    Benzocycloheptenes and heterocyclic analogues as potential drugs. IV. Amines derived from 4-phenyl-8-chloro-2,3,4,5-tetrahydro-1-benzoxepin
    1972, Vol. 37, Issue 6, pp. 2081–2090 [Abstract]
  • Z. Buděšínský and J. Vavřina
    Nucleophilic substitutions in the 2-methanesulfonylpyrimidine series
    1972, Vol. 37, Issue 5, pp. 1721–1733 [Abstract]
  • K. Šindelář, E. Svátek, B. Kakáč, F. Hradil and M. Protiva
    Benzocycloheptenes and heterocyclic analogues as potential drugs. III. Further synthetic experiments in the series of 1-benzothiepin derivatives
    1972, Vol. 37, Issue 4, pp. 1195–1206 [Abstract]
  • Z. Buděšínský, V. Valenta, V. Vosátko and A. Šimek
    Sulfanilamidoquinoxalines
    1972, Vol. 37, Issue 3, pp. 887–895 [Abstract]
  • M. Protiva, V. Seidlová, E. Svátek and F. Hradil
    Benzocycloheptenes and heterocyclic analogues as potential drugs. II. Amines of 8-chloro-2,3,4,5-tetrahydro-1-benzoxepin series
    1972, Vol. 37, Issue 3, pp. 868–886 [Abstract]
  • M. Beran, M. Semonský and E. Svátek
    Substances with antineoplastic activity. XLVII. S-Substituted 6-styryl-3-thioxo-2,3,4,5-tetrahydro-1,2,4-triazin-5-ones and analogous 3-amino(hydrazino) compounds
    1971, Vol. 36, Issue 12, pp. 4000–4005 [Abstract]
  • J. O. Jílek, V. Seidlová, K. Pelz, B. Kakáč, J. Holubek, E. Svátek, Z. Šedivý and M. Protiva
    Neurotropic and psychotropic compounds. XLVIII. Several derivatives of phenanthrene, acenaphthene; anthracene and naphthalene
    1971, Vol. 36, Issue 9, pp. 3300–3313 [Abstract]
  • Z. Buděšínský and A. Valenta
    6,7-Dialkoxychinoxalin-Derivate
    1971, Vol. 36, Issue 7, pp. 2527–2539 [Abstract]
  • O. Exner and E. Svátek
    Substituent effects in infrared spectroscopy. I. The O-H stretching frequencies in monomeric benzoic acids
    1971, Vol. 36, Issue 2, pp. 534–543 [Abstract]
  • V. Zikán, M. Semonský, N. Kucharczyk and E. Svátek
    Substances with antineoplastic activity. XLV. Reduction of β-aroyl-β-halogenoacrylic acids with sodium borohydride
    1970, Vol. 35, Issue 11, pp. 3475–3478 [Abstract]
  • K. Pelz, E. Svátek, J. Metyšová, F. Hradil and M. Protiva
    Neurotropic and psychotropic substances. XLII. 2-Hydroxy-9-(3-dimethylaminopropylidene)thioxanthenes and some related compounds
    1970, Vol. 35, Issue 9, pp. 2623–2634 [Abstract]
  • V. Zikán, M. Semonský and E. Svátek
    Substances with antineoplastic activity. XLIII. Reaction of the ethyl ester of N-(β-4-methoxybenzoyl-β-bromoacryloyl)glycine and -β-alanine with hydrazine; Ethyl ester of N-(β-4-methoxybenzoyl-β-bromoacryloyl)glycylglycine
    1970, Vol. 35, Issue 5, pp. 1434–1439 [Abstract]
  • K. Šindelář, E. Svátek, J. Metyšová, J. Metyš and M. Protiva
    Neurotropic and psychotropic substances. XXXVII. Derivatives of selenoxanthene
    1969, Vol. 34, Issue 12, pp. 3792–3800 [Abstract]
  • K. Šindelář, J. Metyšová, E. Svátek and M. Protiva
    Neurotropic and psychotropic compounds. XXXIV. Derivatives of 6,11-dihydrodibenzo[b,e]selenepin
    1969, Vol. 34, Issue 7, pp. 2122–2127 [Abstract]
  • M. Rajšner, E. Svátek, J. Metyšová and M. Protiva
    Neurotropic and psychotropic compounds. XXXIII. Contribution to the chemistry of 11-(3-dimethylaminopropylidene)-6,11-dihydrodibenzo[b,e]thiepin (prothiadene) and of related compounds
    1969, Vol. 34, Issue 7, pp. 1963–1975 [Abstract]
  • M. Rajšner, E. Svátek, V. Seidlová, E. Adlerová and M. Protiva
    Neurotropic and psychotropic compounds. XXXII. Aminoalkylation of 6,11-dihydrodibenzo[b,e]thiepin 5,5-dioxide and of the corresponding 11-ketone
    1969, Vol. 34, Issue 4, pp. 1278–1285 [Abstract]
  • M. Rajšner, J. Metyš, E. Svátek and M. Protiva
    Neurotropic and psychotropic compounds. XXXI. Chemistry and pharmacology of 11-(3-dimethylaminopropylidene)-2-methyl-6,11-dihydrodibenzo[b,e]thiepin and of some analogues
    1969, Vol. 34, Issue 3, pp. 1015–1024 [Abstract]
  • Z. Buděšínský, J. Přikryl, S. Vaněček and E. Svátek
    Long-acting sulphonamides. IV. Reductive cleavage of the ether bond in the pyrimidine and pyridine series
    1968, Vol. 33, Issue 7, pp. 2266–2275 [Abstract]
  • K. Pelz, V. Seidlová, E. Svátek, M. Rajšner and M. Protiva
    Neurotrope und psychotrope Substanzen XXIV. 2-Substituierte 1,2-Diphenyläthan-Derivate Versuche einer neuen Synthese der Dibenz[b,f]azocin-Derivate
    1968, Vol. 33, Issue 6, pp. 1880–1894 [Abstract]
  • V. Zikán, M. Semonský, E. Svátek and V. Jelínek
    Substanzen mit antineoplastischer Wirkung XIX. Substituierte Pyrazole durch Reaktion von β-4-Methoxybenzoyl-β-chlor(brom)acrylsäure mit Diazomethan
    1967, Vol. 32, Issue 10, pp. 3587–3596 [Abstract]
  • J. O. Jílek, E. Svátek, J. Metyšová, J. Pomykáček and M. Protiva
    Neurotrope und psychotrope Substanzen XVII. 10-(4-Methylpiperazino)-10,11-dihydrodibenzo[b,f]thiepin und einige Analoga
    1967, Vol. 32, Issue 9, pp. 3186–3212 [Abstract]
  • Z. Buděšínský, J. Přikryl and E. Svátek
    2,5-Dihydroxypyrimidine und ihre Derivate
    1967, Vol. 32, Issue 4, pp. 1637–1641 [Abstract]
  • A. Šváb, Z. Buděšínský and J. Vavřina
    Über 5,6-Dihydrofuro[2,3-d]pyrimidine
    1967, Vol. 32, Issue 4, pp. 1582–1587 [Abstract]
  • Z. Buděšínský, J. Přikryl and E. Svátek
    5-Halogenpyrimidine II. Synthese des 2-Hydroxy-5-fluorpyrimidins
    1965, Vol. 30, Issue 11, pp. 3895–3901 [Abstract]
  • J. O. Jílek, J. Pomykáček, E. Svátek, V. Seidlová, M. Rajšner, K. Pelz, B. Hoch and M. Protiva
    Neurotrope und psychotrope Substanzen II. Morphanthridin und Derivate. Neue Synthese des Propazepins
    1965, Vol. 30, Issue 2, pp. 445–462 [Abstract]
  • Z. Buděšínský, J. Přikryl and E. Svátek
    Long-acting sulphonamides. III. New synthesis of 2-sulphanilamido-5-methoxypyrimidine
    1964, Vol. 29, Issue 12, pp. 2980–2991 [Abstract]
  • Z. Buděšínský and F. Roubínek
    In Stellung 4 und 2,4 substituierte 5,6-Tetramethylenpyrimidine
    1964, Vol. 29, Issue 10, pp. 2341–2350 [Abstract]
  • Z. Buděšínský, V. Jelínek and J. Přikryl
    5-Halogenpyrimidine I. Darstellung von 4-Hydroxy-5-halogenpyrimidinen
    1962, Vol. 27, Issue 11, pp. 2550–2560 [Abstract]
  • Z. Buděšínský and F. Roubínek
    Reaktion der Acylbrenztraubensäure-methylester mit Verbindungen vom Harnstoff-Typus
    1961, Vol. 26, Issue 11, pp. 2871–2885 [Abstract]
  • Z. Buděšínský and V. Musil
    Über die Darstellung von 2-Sulfanilamido-4-methylpyrimidinen mit einem heterocyclischen Substituenten in 6-Stellung
    1961, Vol. 26, Issue 11, pp. 2865–2870 [Abstract]
  • L. Macholán and E. Svátek
    Aminoketocarbonsäuren VI. Über die Konstitution und Strukturformen der α-Ketoanaloga natürlicher Diaminosäuren
    1960, Vol. 25, Issue 10, pp. 2564–2574 [Abstract]
  • Z. Buděšínský and V. Musil
    Darstellung der 2-Sulfanilamido-4-methyl-6-alkylpyrimidine
    1959, Vol. 24, Issue 12, pp. 4022–4028 [Abstract]
  • R. Zahradník, E. Svátek and M. Chvapil
    Nitrosamine sekundärer Amine III. Spektroskopische und polarographische Studie
    1959, Vol. 24, Issue 2, pp. 347–359 [Abstract]
  • Z. Buděšínský and A. Šváb
    Über die Synthese von Äthylestern und Amiden substituierter 1,3-Dihydroxynaphthalin-2-carbonsäuren
    1958, Vol. 23, Issue 6, pp. 1066–1071 [Abstract]
  • Z. Buděšínský and A. Šváb
    Antituberkulose Substanzen XIII. Darstellung von 3-Amino-4-alkoxy-propenylbenzolen
    1957, Vol. 22, Issue 5, pp. 1645–1648 [Abstract]
  • Z. Buděšínský and E. Ročková
    Antituberkulöse Stoffe XII. Imidazolid-2-thion-4-carbonsäuren
    1957, Vol. 22, Issue 3, pp. 811–815 [Abstract]
  • A. Emr and F. Roubínek
    Synthese der Thioäpfelsäure
    1956, Vol. 21, Issue 6, pp. 1651–1653 [Abstract]
  • E. Knobloch and E. Svátek
    Polarographie des Chloramphenikols und verwandter Stoffe
    1955, Vol. 20, Issue 5, pp. 1113–1124 [Abstract]
  • Z. Buděšínský and J. Kopecký
    Eine neue Synthese der Pyrimidinkomponente des Vitamins B1
    1955, Vol. 20, Issue 1, pp. 52–58 [Abstract]
  • Z. Buděšínský and E. Ročková
    Antituberculous compounds. IX. Some allyl- and propenyl- derivatives of m-aminophenol
    1954, Vol. 19, Issue 5, pp. 966–975 [Abstract]
  • Z. Buděšínský and A. Šváb
    Antituberculous compounds. VIII. Preparation of 2-carboxy- and 2-aminoanethole
    1954, Vol. 19, Issue 5, pp. 959–965 [Abstract]
  • E. Svátek, Z. Roubal and R. Přibil
    New complex-forming compounds in polarography. II. Pyrocatechol-3,5-disulphonic acid
    1954, Vol. 19, Issue 4, pp. 674–678 [Abstract]
  • R. Přibil, Z. Roubal and E. Svátek
    New complex-forming reagents in polarography. I. 1,2-Diaminocyclohexane-N,N,N',N'-tetra-acetic acid
    1953, Vol. 18, Issue 1, pp. 43–52 [Abstract]
  • Z. Buděšínský and J. Šolín
    On the preparation of certain new asymmetric sulfones
    1949, Vol. 14, pp. 267–273 [Abstract]
  • Z. Buděšínský
    On some new derivatives of 2-methylpyrimidine
    1949, Vol. 14, pp. 223–235 [Abstract]