Collect. Czech. Chem. Commun.
1980, 45, 135-141
https://doi.org/10.1135/cccc19800135
Reactions and spectral properties of ethyl 5-aminofuroate and its derivatives
Josef Prousek, Adolf Jurášek and Jaroslav Kováč
Department of Organic Chemistry, Slovak Institute of Technology, 880 37 Bratislava
Abstract
Ethyl 5-aminofuroate (II), prepared by reduction of ethyl 5-nitrofuroate (I), served for preparation of bifunctional α,β-substituted aminofurans IV-IX, acyl derivatives IIIa, IIIb and condensation product X. The latter reacted with diazomethane directly to afford the corresponding aziridine derivative XI. The synthesized compounds were characterized by spectral data (IR, UV, 1H-NMR, 13C-NMR (XI) and mass spectra.)
