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Collect. Czech. Chem. Commun. 2000, 65, 280-296
https://doi.org/10.1135/cccc20000280

Synthesis and Analgesic Activity of Some 1-Benzofurans, 1-Benzothiophenes and Indoles

Stanislav Rádla,*, Petr Hezkýa, Jitka Urbánkováb, Petr Váchalb and Ivan Krejčía

a Research Institute of Pharmacy and Biochemistry, Kouřimská 17, 130 60 Prague 3, Czech Republic
b Department of Organic Chemistry, Prague Institute of Chemical Technology, 166 28 Prague 6, Czech Republic

Crossref Cited-by Linking

  • Diao Peng-Cheng, Hu Meng-Jin, Yang Hai-Kui, You Wen-Wei, Zhao Pei-Liang: Facile one-pot synthesis, antiproliferative evaluation and structure-activity relationships of 3-amino-1H-indoles and 3-amino-1H-7-azaindoles. Bioorganic Chemistry 2019, 88, 102914. <https://doi.org/10.1016/j.bioorg.2019.04.008>
  • Sayed Mostafa, Kamal El-Dean Adel M., Ahmed Mostafa, Hassanien Reda: Synthesis of some heterocyclic compounds derived from indole as antimicrobial agents. Synthetic Communications 2018, 48, 413. <https://doi.org/10.1080/00397911.2017.1403627>
  • Demidov Maxim R., Lapshina Marina Yu., Osipov Dmitry V., Osyanin Vitaly A., Klimochkin Yuri N.: Oxidative rearrangement of 4H-chromenes to 2-aroylbenzofurans in the presence of selenium dioxide. Chem Heterocycl Comp 2017. <https://doi.org/10.1007/s10593-017-2169-7>
  • Anantacharya R., Manjulatha K., Satyanarayan N.D., Santoshkumar S., Kaviraj M.Y., Spencer John: Antiproliferative, DNA cleavage, and ADMET study of substituted 2-(1-benzofuran-2-yl) quinoline-4-carboxylic acid and its esters. Cogent Chemistry 2016, 2, 1158382. <https://doi.org/10.1080/23312009.2016.1158382>
  • Shakya Ashok K., Kamal Mehnaz, Balaramnavar Vishal M., Bardaweel Sanna K., Naik Rajashri R., Saxena Anil K., Siddiqui H. H.: Design, synthesis and evaluation of benzofuran-acetamide scaffold as potential anticonvulsant agent. Acta Pharmaceutica 2016, 66. <https://doi.org/10.1515/acph-2016-0023>
  • Senadi Gopal Chandru, Hu Wan-Ping, Boominathan Siva Senthil Kumar, Wang Jeh-Jeng: Palladium(0)-Catalyzed Single and Double Isonitrile Insertion: A Facile Synthesis of Benzofurans, Indoles, and Isatins. Chem. Eur. J. 2015, 21, 998. <https://doi.org/10.1002/chem.201405933>
  • Aswathanarayanappa Chandrashekar, Bheemappa Eswarappa, Bodke Yadav D., Bhovi Venkatesh K., Ningegowda Raghu, Shivakumar M. C., Peethambar S. K., Telkar Sandeep: 5-phenyl-1-benzofuran-2-yl derivatives: synthesis, antimicrobial, and antioxidant activity. Med Chem Res 2013, 22, 78. <https://doi.org/10.1007/s00044-012-0017-y>
  • Rokade Balaji V., Prabhu Kandikere Ramaiah: Chemoselective Schmidt Reaction Mediated by Triflic Acid: Selective Synthesis of Nitriles from Aldehydes. J. Org. Chem. 2012, 77, 5364. <https://doi.org/10.1021/jo3008258>
  • Abdel-Rahman Adel A.H., El-Latif Mona M. Abd, El-Essawy Farag A., Barakat Yousif A.: Synthesis and Antiviral Activity of 3-Aminoindole Nucleosides of 2-Acetamido-2-deoxy-D-glucose. Bulletin of the Korean Chemical Society 2012, 33, 3417. <https://doi.org/10.5012/bkcs.2012.33.10.3417>
  • Trivedi Amit R., Desai Jignesh M., Dholariya Bipin H., Dodiya Dipti K., Shah Viresh H.: Synthesis and antimicrobial evaluation of novel benzo[b]thiophenes comprising β-lactam nucleus. Med Chem Res 2011, 21, 1471. <https://doi.org/10.1007/s00044-011-9669-2>
  • Radl Stanislav, Hezky Petr, Urbankova Jitka, Vachal Petr, Krejci Ivan: ChemInform Abstract: Synthesis and Analgesic Activity of Some 1-Benzofurans, 1-Benzothiophenes and Indoles. ChemInform 2010, 31, no. <https://doi.org/10.1002/chin.200028043>
  • Velezheva V.S., Azev V.N., Kornienko A.G., Peregudov A.S., Godovikov I.A., Sebyakin Yu. L.: The stereoselective synthesis of highly functionalized tertiary 3-aminoindoles/anilines or dihydropyrroles from C-(3-indolyl)-N-aryl and C,N-diaryl nitrones. Tetrahetron Lett 2010, 51, 6594. <https://doi.org/10.1016/j.tetlet.2010.10.045>
  • Seong Churl Min, Park Chul Min, Choi Jinil, Park No Sang: An efficient base-mediated intramolecular condensation of 2-(disubstituted amino)-benzonitriles to 3-aminoindoles. Tetrahetron Lett 2009, 50, 1029. <https://doi.org/10.1016/j.tetlet.2008.12.052>
  • Romagnoli Romeo, Baraldi Pier Giovanni, Jung M. Katherine, Iaconinoto Maria Antonietta, Carrion Maria Dora, Remusat Vincent, Preti Delia, Tabrizi Mojgan Aghazadeh, Francesca Fruttarolo, De Clercq Erik: Synthesis and preliminary biological evaluation of new anti-tubulin agents containing different benzoheterocycles. Biorg Med Chem Lett 2005, 15, 4048. <https://doi.org/10.1016/j.bmcl.2005.06.022>
  • Ando Kumiko, Tsuji Eriko, Ando Yuko, Kuwata Noriko, Kunitomo Jun-ichi, Yamashita Masayuki, Ohta Shunsaku, Kohno Shigekatsu, Ohishi Yoshitaka: Syntheses of 3-acetoacetylaminobenzo[b]furan derivatives having cysteinyl leukotriene 2 receptor antagonistic activity. Org. Biomol. Chem. 2004, 2, 625. <https://doi.org/10.1039/B312682J>
  • Nettekoven Matthias: Combinatorial synthesis of libraries of indole derivatives. Biorg Med Chem Lett 2001, 11, 2169. <https://doi.org/10.1016/S0960-894X(01)00393-6>
  • Rádl Stanislav, Konvička Petr, Váchal Petr: A new approach to the synthesis of benzofuro[3,2-b]quinolines, benzothieno[3,2-b]quinolines and indolo[3,2-b]quinolines. Journal of Heterocyclic Chemistry 2000, 37, 855. <https://doi.org/10.1002/jhet.5570370430>
  • Rádl Stanislav, Hezký Petr, Konvička Petr, Krejčí Ivan: Synthesis and Analgesic Activity of Some Substituted 1-Benzofurans and 1-Benzothiophenes. Collect. Czech. Chem. Commun. 2000, 65, 1093. <https://doi.org/10.1135/cccc20001093>