Crossref Cited-by Linking logo

Collect. Czech. Chem. Commun. 1986, 51, 2802-2809
https://doi.org/10.1135/cccc19862802

Some nucleophilic reactions of 2-isothiocyanatobenzyl bromide. A new simple synthesis of 2-substituted 4H-benzo[d][1,3]thiazines

Jozef Gonda and Pavol Kristian

Department of Organic Chemistry and Biochemistry, faculty of Natural Sciences, P. J. Šafárik University, 041 67 Košice

Crossref Cited-by Linking

  • Hassanzadeh Leila, Chen Suxiang, Veedu Rakesh: Radiolabeling of Nucleic Acid Aptamers for Highly Sensitive Disease-Specific Molecular Imaging. Pharmaceuticals 2018, 11, 106. <https://doi.org/10.3390/ph11040106>
  • Jun Hee‐Goo, Kim Eun‐Mi, Yoon Hyo‐Jeong, Gong Young‐Dae: Microwave‐assisted Solid‐phase Synthesis of N‐substituted‐2‐aminobenzo[d][1,3] Thiazine Derivatives from a BOMBA Resin. Bulletin Korean Chem Soc 2017, 38, 334. <https://doi.org/10.1002/bkcs.11088>
  • Kobayashi Kazuhiro, Nogi Takashi: Synthesis of 2-Alk(or Aryl)oxy- and 2-(Alkyl(or Aryl)sulfanyl)-4H-3,1-benzothiazine Derivatives Carrying a (Z)-Halomethylidene Substutuent at the 4-Position. HETEROCYCLES 2016, 92, 1810. <https://doi.org/10.3987/COM-16-13530>
  • Hua Lu, Yao Zhigang, Xu Fan, Shen Qi: Chemoselective reactions under solvent-free conditions: lanthanide-catalyzed syntheses of 2-amino-3,1-benzothiazines and 3,4-dihydroquinazoline-2-thiones. RSC Adv. 2014, 4, 3113. <https://doi.org/10.1039/C3RA44829K>
  • Pandey Garima, Bhowmik Subhendu, Batra Sanjay: Synthesis of 4-substituted imino-4H-benzo[d][1,3] thiazin-2-amines via palladium-catalysed isocyanide insertion in 2-bromophenylthioureas. RSC Adv. 2014, 4, 41433. <https://doi.org/10.1039/C4RA06875K>
  • Huang Jie, Yu Yong, Hua Lu, Yao ZhiGang, Xu Fan, Shen Qi: Tandem addition-cyclization reaction catalyzed by ytterbium chloride: An efficient one-step synthesis of 2-amino-4H-3,1-benzothiazine. Chin. Sci. Bull. 2013, 58, 717. <https://doi.org/10.1007/s11434-012-5631-z>
  • Kobayashi Kazuhiro, Ezaki Kosuke, Tanmatsu Miyuki: Synthesis of 2-Sulfanyl-4H-3,1-benzothiazine Derivatives by the Reaction of 2-(Bromomethyl)phenyl Isothiocyanates with Thiols. HETEROCYCLES 2013, 87, 1311. <https://doi.org/10.3987/COM-13-12701>
  • Kobayashi Kazuhiro, Ezaki Kosuke: One-Pot Synthesis of 2-(1,4-Dihydro-2H-3,1-benzothiazin-2-ylidene)propanedioic Acid Derivatives by the Reaction of 2-(1-Bromoalkyl)phenyl Isothiocyanates with Propanedioic Acid Derivatives Using Sodium Hydride. HETEROCYCLES 2012, 85, 3007. <https://doi.org/10.3987/COM-12-12584>
  • Kobayashi Kazuhiro, Kanbe Yuuki: Two-pot synthesis of N,N-disubstituted 4H-3,1-benzothiazin-2-amines from aryl(2-isothiocyanatophenyl)methanones and secondary amines. Tedrahedron 2011, 67, 9680. <https://doi.org/10.1016/j.tet.2011.10.045>
  • Otani Takashi, Katsurayama Saki, Ote Tatsuya, Saito Takao: Stereoselective synthesis of 4H-3,1-benzothiazines via tandem nucleophilic addition/epoxy ring-opening cyclization reactions of 2-(3-phenyloxiranyl)phenyl isothiocyanates. Journal of Sulfur Chemistry 2009, 30, 250. <https://doi.org/10.1080/17415990902839443>
  • Fedotov A. N., Trofimova E. V., Romanov V. A., Mochalov S. S., Shabarov Yu. S., Zefirov N. S.: Synthesis of 2-amino-4H-3,1-benzoxazines and 2-amino-4H-3,1-benzothiazines by the rearrangement of o-cyclopropylphenylureas and o-cyclopropylphenylthioureas. Chem Heterocycl Comp 2008, 44, 96. <https://doi.org/10.1007/s10593-008-0006-8>
  • Fedotov A. N., Trofimova E. V., Sidorov V. A., Potekhin K. A., Romanov V. A., Mochalov S. S., Zefirov N. S.: 2-Amino-4H-3,1-benzothiazines from Arylcyclopropanes: Crystal Structure of the Product of N1-(2-Cyclopropylphenyl)-N2-(2-ethylphenyl)thiourea Rearrangement. Dokl Chem 2005, 405, 217. <https://doi.org/10.1007/s10631-005-0076-4>
  • Lobodin Vladislav V., Fedotov Alexandr N., Dem’yanov Piotr I., Lebedev Albert T., Ovcharenko Vladimir V., Pihlaja Kalevi, Blumenthal Tom: Cyclization of the substituted N-(Ortho-cyclopropylphenyl)-N′-aryl ureas and thioureas in the gas phase and solution. J. Am. Soc. Mass Spectrom. 2005, 16, 1739. <https://doi.org/10.1016/j.jasms.2005.07.006>
  • Maligres Peter E., Waters Marjorie S., Weissman Steven A., McWilliams J. Christopher, Lewis Stephanie, Cowen Jennifer, Reamer Robert A., Volante R. P., Reider Paul J., Askin David: Preparation of a clinically investigated ras farnesyl transferase inhibitor. Journal of Heterocyclic Chem 2003, 40, 229. <https://doi.org/10.1002/jhet.5570400206>
  • Litak Peter T., Kauffman Joel M.: Syntheses of reactive fluorescent stains derived from 5(2)‐aryl‐2(5)‐(4‐pyridyl)oxazoles and bifunctionally reactive linkers. Journal of Heterocyclic Chem 1994, 31, 457. <https://doi.org/10.1002/jhet.5570310236>
  • Lee Hyunil, Kim Kyongtae: A facile synthesis of 2‐cyano‐4H‐3,1‐ benzothiazines and 2‐cyano‐4H‐3,1‐benzoxazines. Heteroatom Chemistry 1993, 4, 263. <https://doi.org/10.1002/hc.520040222>
  • GONDA J., KRISTIAN P.: ChemInform Abstract: Some Nucleophilic Reactions of 2‐Isothiocyanatobenzyl Bromide. A New Simple Synthesis of 2‐Substituted 4H‐Benzo(d) (1,3)thiazines. ChemInform 1987, 18. <https://doi.org/10.1002/chin.198718230>