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Collect. Czech. Chem. Commun. 1986, 51, 2802-2809
https://doi.org/10.1135/cccc19862802

Some nucleophilic reactions of 2-isothiocyanatobenzyl bromide. A new simple synthesis of 2-substituted 4H-benzo[d][1,3]thiazines

Jozef Gonda and Pavol Kristian

Department of Organic Chemistry and Biochemistry, faculty of Natural Sciences, P. J. Šafárik University, 041 67 Košice

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  • Kobayashi Kazuhiro, Nogi Takashi: Synthesis of 2-Alk(or Aryl)oxy- and 2-(Alkyl(or Aryl)sulfanyl)-4H-3,1-benzothiazine Derivatives Carrying a (Z)-Halomethylidene Substutuent at the 4-Position. HETEROCYCLES 2016, 92, 1810. <https://doi.org/10.3987/COM-16-13530>
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  • Kobayashi Kazuhiro, Ezaki Kosuke, Tanmatsu Miyuki: Synthesis of 2-Sulfanyl-4H-3,1-benzothiazine Derivatives by the Reaction of 2-(Bromomethyl)phenyl Isothiocyanates with Thiols. HETEROCYCLES 2013, 87, 1311. <https://doi.org/10.3987/COM-13-12701>
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  • Fedotov A. N., Trofimova E. V., Romanov V. A., Mochalov S. S., Shabarov Yu. S., Zefirov N. S.: Synthesis of 2-amino-4H-3,1-benzoxazines and 2-amino-4H-3,1-benzothiazines by the rearrangement of o-cyclopropylphenylureas and o-cyclopropylphenylthioureas. Chem Heterocycl Comp 2008, 44, 96. <https://doi.org/10.1007/s10593-008-0006-8>
  • Fedotov A. N., Trofimova E. V., Sidorov V. A., Potekhin K. A., Romanov V. A., Mochalov S. S., Zefirov N. S.: 2-Amino-4H-3,1-benzothiazines from Arylcyclopropanes: Crystal Structure of the Product of N1-(2-Cyclopropylphenyl)-N2-(2-ethylphenyl)thiourea Rearrangement. Dokl Chem 2005, 405, 217. <https://doi.org/10.1007/s10631-005-0076-4>
  • Lobodin Vladislav V., Fedotov Alexandr N., Dem’yanov Piotr I., Lebedev Albert T., Ovcharenko Vladimir V., Pihlaja Kalevi, Blumenthal Tom: Cyclization of the substituted N-(Ortho-cyclopropylphenyl)-N′-aryl ureas and thioureas in the gas phase and solution. j am soc mass spectrom 2005, 16, 1739. <https://doi.org/10.1016/j.jasms.2005.07.006>
  • Maligres Peter E., Waters Marjorie S., Weissman Steven A., McWilliams J. Christopher, Lewis Stephanie, Cowen Jennifer, Reamer Robert A., Volante R. P., Reider Paul J., Askin David: Preparation of a clinically investigated ras farnesyl transferase inhibitor. Journal of Heterocyclic Chemistry 2003, 40, 229. <https://doi.org/10.1002/jhet.5570400206>
  • Litak Peter T., Kauffman Joel M.: Syntheses of reactive fluorescent stains derived from 5(2)-aryl-2(5)-(4-pyridyl)oxazoles and bifunctionally reactive linkers. Journal of Heterocyclic Chemistry 1994, 31, 457. <https://doi.org/10.1002/jhet.5570310236>
  • Lee Hyunil, Kim Kyongtae: A facile synthesis of 2-cyano-4H-3,1- benzothiazines and 2-cyano-4H-3,1-benzoxazines. Heteroat. Chem. 1993, 4, 263. <https://doi.org/10.1002/hc.520040222>
  • GONDA J., KRISTIAN P.: ChemInform Abstract: Some Nucleophilic Reactions of 2-Isothiocyanatobenzyl Bromide. A New Simple Synthesis of 2-Substituted 4H-Benzo(d) (1,3)thiazines. ChemInform 1987, 18. <https://doi.org/10.1002/chin.198718230>